SCHEMBL10488186

SCHEMBL10488186

CCCCS(=O)(=O)Nc1ccc(CCCCOCCCCCCNCc2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.52
SIGMAR1 Q99720 3/20 0.50
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
S1PR1 P21453 7/20 0.46
S1PR3 Q99500 7/20 0.46
S1PR2 O95136 5/20 0.46
S1PR4 O95977 3/20 0.45
HPGD P15428 2/20 0.45
BCHE P06276 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
LPAR2 Q9HBW0 2/20 0.43
S1PR5 Q9H228 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
CA12 O43570 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10477677 0.98 AR (0.52) ARSIGMAR1CNR1CNR2S1PR1
SCHEMBL9762923 0.96 AR (0.52) ARSIGMAR1CNR1CNR2S1PR1
SCHEMBL9763021 0.86 AR (0.51) ARSIGMAR1CNR1CNR2S1PR1
SCHEMBL9762627 0.83 SIGMAR1 (0.52) ARSIGMAR1CNR1CNR2S1PR1
SCHEMBL9763280 0.83 SIGMAR1 (0.55) ARSIGMAR1BCHEALDH1A1MEN1
SCHEMBL9763725 0.81 DRD2 (0.51) ARSIGMAR1HPGDBCHEALDH1A1
SCHEMBL10463959 0.81 HPGD (0.50) ARHPGDLMNAADRB2ADRB1
SCHEMBL456614 0.79 SIGMAR1 (0.80) SIGMAR1CNR1CNR2BCHE
SCHEMBL10477931 0.79 HPGD (0.50) ARHPGDLMNAADRB2ADRB1
Bromide SCHEMBL7121198 0.78 SIGMAR1 (0.77) SIGMAR1CNR1CNR2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4853382-A TREATING ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1989-08-01 US disclosed
EP-0178919-B1 AMINOPHENOL DERIVATIVES GLAXO GROUP LIMITED (GB) 1988-12-21 EP disclosed
US-4730008-A STIMULANT FOR BETA-ADRENORECEPTORS GLAXO GROUP LIMITED (GB) 1988-03-08 US disclosed