SCHEMBL9763725

SCHEMBL9763725

CS(=O)(=O)Nc1ccc(CCOCCCCCCNCc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.51
DRD3 P35462 2/20 0.51
DRD4 P21917 1/20 0.51
SIGMAR1 Q99720 3/20 0.49
ADRB2 P07550 2/20 0.47
ADRB1 P08588 2/20 0.47
ADRB3 P13945 2/20 0.47
MAOA P21397 1/20 0.47
CHRM2 P08172 1/20 0.46
HPGD P15428 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
AR P10275 1/20 0.45
RAB9A P51151 1/20 0.45
BCHE P06276 2/20 0.43
GRIN1 Q05586 1/20 0.42
KCNH2 Q12809 1/20 0.42
GRIN2B Q13224 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7907015 0.86 SIGMAR1 (0.64) DRD2DRD3DRD4SIGMAR1ADRB2
SCHEMBL9762923 0.86 AR (0.52) SIGMAR1ADRB2ADRB1ADRB3MAOA
SCHEMBL9764394 0.83 SIGMAR1 (0.69) SIGMAR1MAOACHRM2BCHE
SCHEMBL10477755 0.83 SIGMAR1 (0.69) SIGMAR1MAOACHRM2BCHE
SCHEMBL9762627 0.83 SIGMAR1 (0.52) SIGMAR1ADRB3MAOACHRM2HPGD
SCHEMBL9763280 0.83 SIGMAR1 (0.55) SIGMAR1ADRB1ADRB3MAOACHRM2
Hydrochloric Acid SCHEMBL9258435 0.82 SIGMAR1 (0.67) SIGMAR1MAOACHRM2BCHE
SCHEMBL9763689 0.82 SIGMAR1 (0.52) SIGMAR1MAOACHRM2BCHE
SCHEMBL9763494 0.81 DRD2 (0.47) DRD2DRD3DRD4SIGMAR1ADRB2
SCHEMBL10488186 0.81 AR (0.52) SIGMAR1ADRB2ADRB1ADRB3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4990505-A Treating asthma, bronchitis; adrenergic stimulants GLAXO GROUP LIMITED (GB) 1991-02-05 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed