SCHEMBL10501484

SCHEMBL10501484

CSc1ccc(Oc2ccc(N3NCC(=O)NC3=O)cc2)cc1C

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.43
SLC6A4 P31645 7/20 0.37
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
HSD17B10 Q99714 1/20 0.36
SLC6A2 P23975 4/20 0.33
SLC6A3 Q01959 4/20 0.33
HRH3 Q9Y5N1 4/20 0.33
HPGD P15428 1/20 0.33
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
EIF2AK2 P19525 1/20 0.31
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9502409 0.85 THRB (0.44) THRBSLC6A4ALDH1A1CYP3A4TSHR
SCHEMBL9500876 0.76 THRB (0.38) THRBSLC6A4SLC6A2SLC6A3RAB9A
SCHEMBL10501699 0.71 SLC6A4 (0.40) SLC6A4SLC6A2SLC6A3HRH3MEN1
SCHEMBL9504425 0.71 NPBWR1 (0.35) SLC6A4ALDH1A1SLC6A2SLC6A3RAB9A
SCHEMBL10502467 0.70 NPC1 (0.40) ALDH1A1TSHRMAPTRAB9A
SCHEMBL10501494 0.69 KMT2A (0.36) ALDH1A1CYP3A4TSHRHPGDMEN1
SCHEMBL11452562 0.68 THRB (0.80) THRBSLC6A4
SCHEMBL11661452 0.67 CYP3A4 (0.49) THRBSLC6A4ALDH1A1CYP3A4TSHR
SCHEMBL11455388 0.67 ALDH1A1 (0.53) THRBSLC6A4ALDH1A1CYP3A4TSHR
SCHEMBL11456434 0.65 L3MBTL1 (0.50) THRBSLC6A4ALDH1A1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154885-B1 SUBSTITUTED 2-PHENYL-HEXAHYDRO-1,2,4-TRIAZINE-2,5-DIONES, METHOD FOR THEIR PREPARATION, THEIR USE AS VETERINARY MEDICINES AND FOR COMBATING PROTOZOES HOECHST AKTIENGESELLSCHAFT (DE) 1989-01-18 EP disclosed
US-4640917-A 2-phenyl-hexahydro-1,2,4-triazine-3,5-diones HOECHST AKTIENGESELLSCHAFT (DE) 1987-02-03 US disclosed
EP-0154885-A1 Substituted 2-phenyl-hexahydro-1,2,4-triazine-2,5-diones, method for their preparation, their use as veterinary medicines and for combating protozoes HOECHST AKTIENGESELLSCHAFT (DE) 1985-09-18 EP disclosed