SCHEMBL10502467

SCHEMBL10502467

CSc1ccc(Sc2ccc(N3NCC(=O)NC3=O)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PTGS2 P35354 2/20 0.33
ALDH1A1 P00352 4/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
GSK3B P49841 1/20 0.32
PSMB2 P49721 1/20 0.31
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10501019 0.86 MAOA (0.41) NPC1RAB9AALDH1A1LMNAGSK3B
SCHEMBL10501494 0.83 KMT2A (0.36) NPC1ALDH1A1SMN1; SMN2MAPTTSHR
SCHEMBL9501160 0.83 LMNA (0.36) NPC1RAB9AALDH1A1SMN1; SMN2LMNA
SCHEMBL9500876 0.75 THRB (0.38) NPC1RAB9APTGS2
SCHEMBL9504425 0.74 NPBWR1 (0.35) NPC1RAB9APTGS2ALDH1A1SMN1; SMN2
SCHEMBL6248177 0.73 DDB1 (0.47) NPC1RAB9APTGS2ALDH1A1LMNA
SCHEMBL10733171 0.72 HTR1A (0.36) PTGS2ALDH1A1MAPT
SCHEMBL9504429 0.72 MEN1 (0.38) LMNAMAPK1MAPT
SCHEMBL9501084 0.71 MEN1 (0.42) LMNAMAPK1MAPT
SCHEMBL9502415 0.67 KMT2A (0.34) ALDH1A1SMN1; SMN2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154885-B1 SUBSTITUTED 2-PHENYL-HEXAHYDRO-1,2,4-TRIAZINE-2,5-DIONES, METHOD FOR THEIR PREPARATION, THEIR USE AS VETERINARY MEDICINES AND FOR COMBATING PROTOZOES HOECHST AKTIENGESELLSCHAFT (DE) 1989-01-18 EP disclosed
US-4640917-A 2-phenyl-hexahydro-1,2,4-triazine-3,5-diones HOECHST AKTIENGESELLSCHAFT (DE) 1987-02-03 US disclosed
EP-0154885-A1 Substituted 2-phenyl-hexahydro-1,2,4-triazine-2,5-diones, method for their preparation, their use as veterinary medicines and for combating protozoes HOECHST AKTIENGESELLSCHAFT (DE) 1985-09-18 EP disclosed