SCHEMBL10547366

SCHEMBL10547366

COc1cc(Br)c([C@@H]2C=C[C@H](c3c(Br)cc(OC)cc3Br)C2)c(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
GRM2 Q14416 1/20 0.34
MAOA P21397 2/20 0.33
MAOB P27338 2/20 0.33
CYP1A1 P04798 1/20 0.32
CYP1B1 Q16678 1/20 0.32
CYP3A4 P08684 1/20 0.31
KDM1A O60341 1/20 0.31
CA2 P00918 1/20 0.30
CA4 P22748 1/20 0.30
TSHR P16473 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26207348 0.67 MAOA (0.37) ALDH1A1GRM2MAOAMAOBHTR2A
SCHEMBL1012684 0.66 HSD17B10 (0.31) MAOAMAOBKDM1A
SCHEMBL11403757 0.66 ALDH1A1 (0.59) ALDH1A1CYP1A1CYP1B1CYP3A4CA2
SCHEMBL11526269 0.65 CHRNB2 (0.41) CYP1A1CYP1B1CYP3A4CA2HTR2A
SCHEMBL4402559 0.65 MTNR1A (0.43) HTR2AHTR2C
SCHEMBL25429872 0.64 MEN1 (0.41) MAOAMAOBHTR2AHTR2C
SCHEMBL30550467 0.64 MAOA (0.40) MAOAMAOBCA2
SCHEMBL1119927 0.64 CA2 (0.56) ALDH1A1CYP1A1CYP1B1CYP3A4CA2
SCHEMBL4297601 0.64 ALDH1A1 (0.56) ALDH1A1CYP1A1CYP1B1CYP3A4CA2
SCHEMBL31562352 0.63 CYP3A4 (0.41) ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4822804-A 5,6,7,-trinor-4,8-inter-m-phenylene 2-nor PGI2 derivatives and anti-ulcer, anti-thrombotic and anti-hypertensive pharmaceutical compositions containing them TORAY INDUSTRIES, INC. (JP) 1989-04-18 US disclosed
US-4564620-A 5,6,7,-Trinor-4,8-inter-m-phenylene PGI2 derivatives and anti-ulcer, anti-thrombotic and anti-hypertensive pharmaceutical compositions containing them TORAY INDUSTRIES, INC. (JP) 1986-01-14 US disclosed