SCHEMBL10594957

SCHEMBL10594957

COC(=O)CCSc1cnns1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.40
CXCR1 P25024 1/20 0.38
CXCR2 P25025 1/20 0.38
GSTP1 P09211 1/20 0.37
GSTM2 P28161 1/20 0.37
TSHR P16473 2/20 0.36
HSD17B10 Q99714 3/20 0.35
ALDH1A1 P00352 4/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
APP P05067 1/20 0.33
POLB P06746 2/20 0.33
MEN1 O00255 1/20 0.33
RAB9A P51151 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10818255 0.85 ALDH1A1 (0.46) TSHRHSD17B10ALDH1A1KMT2AMAPT
SCHEMBL9627350 0.75 PTGS1 (0.40) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL970491 0.74 PTGS1 (0.39) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL10404352 0.73 SMN1; SMN2 (0.35) ALDH1A1KMT2AMAPTLMNAHTT
SCHEMBL16724105 0.73 SMN1; SMN2 (0.41) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL21963005 0.70 CCNE2 (0.44) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL10402932 0.69 RPS6KA3 (0.33)
SCHEMBL9097022 0.69 CA2 (0.45) PTGS1CXCR1CXCR2HSD17B10
SCHEMBL23569353 0.68 CXCR1 (0.40) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL15315500 0.67 RAB9A (0.46) PTGS1CXCR1CXCR2TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0104403-B1 NEW METHOD FOR THE SYNTHESIS OF 5-THIO-1,2,3-THIADIAZOLE AMERICAN CYANAMID COMPANY (US) 1989-01-25 EP disclosed
US-4454336-A Derivatives of 3-(formylmethylthio)-propanoate AMERICAN CYANAMID COMPANY (US) 1984-06-12 US disclosed
EP-0104403-A1 New method for the synthesis of 5-thio-1,2,3-thiadiazole AMERICAN CYANAMID COMPANY (US) 1984-04-04 EP disclosed