SCHEMBL10654899

SCHEMBL10654899

CS(=O)(=O)c1scc(-c2cccc(F)c2)c1C#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
HPGD P15428 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
KDR P35968 1/20 0.39
ADORA2B P29275 2/20 0.39
ADORA1 P30542 2/20 0.39
SLC22A12 Q96S37 1/20 0.39
KMT2A Q03164 2/20 0.39
ADORA2A P29274 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
IDO1 P14902 1/20 0.37
PTGS2 P35354 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10653342 0.84 ATM (0.51) KDM4EHPGDNPSR1ADORA2BADORA1
SCHEMBL10656112 0.83 ALDH1A1 (0.50) KDM4EHPGDNPSR1ADORA1KMT2A
SCHEMBL10653380 0.80 GRIA2 (0.33) KDM4EHPGDNPSR1KMT2AALDH1A1
SCHEMBL10653117 0.77 ABL1 (0.40) ADORA1ADORA2AIDO1PTGS2PRKCZ
SCHEMBL10651486 0.75 PTGS2 (0.43) KDM4EHPGDNPSR1RXFP1KMT2A
SCHEMBL10652386 0.75 GRIA2 (0.42) SLC22A12KMT2AALDH1A1SMN1; SMN2PTGS2
SCHEMBL10656208 0.73 NPSR1 (0.50) KDM4EHPGDNPSR1RXFP1ADORA1
SCHEMBL10651545 0.71 HSP90AA1 (0.40) KDM4EHPGDNPSR1RXFP1ADORA1
SCHEMBL10651866 0.69 KDM4E (0.47) KDM4EHPGDNPSR1KDRKMT2A
SCHEMBL24910100 0.68 ACLY (0.44) KDM4EHPGDNPSR1RXFP1SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273602-A1 3-Cyano-4-arylthiophenes ELI LILLY AND COMPANY (US) 1988-07-06 EP disclosed