SCHEMBL10669673

SCHEMBL10669673

C=CCn1nc(C)c(NCCNCC(O)c2ccc(O)cc2)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 4/20 0.38
ALDH1A1 P00352 3/20 0.38
TAAR1 Q96RJ0 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HTR1A P08908 1/20 0.38
THPO P40225 1/20 0.38
BLM P54132 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NMUR2 Q9GZQ4 1/20 0.38
CYP2C9 P11712 1/20 0.38
ADRB2 P07550 5/20 0.37
CYP3A4 P08684 2/20 0.37
TSHR P16473 2/20 0.37
NFKB1 P19838 2/20 0.37
LMNA P02545 2/20 0.37
ADRB1 P08588 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
SLC22A1 O15245 1/20 0.37
CHRM2 P08172 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10671458 0.90 CYP2D6 (0.43) ALDH1A1TDP1KDM4ESMN1; SMN2ADRB2
SCHEMBL10670001 0.89 HIF1A (0.47) HIF1AKDM4EHTR1ABLMADRB2
SCHEMBL10669677 0.80 ADRB2 (0.30) HIF1AADRB2LMNAADRB1SLC6A4
SCHEMBL10569784 0.75 MEN1 (0.46) CYP2C9ADRB2CYP3A4TSHRLMNA
SCHEMBL10670257 0.74 LMNA (0.48) ALDH1A1KDM4EADRB2CYP3A4LMNA
SCHEMBL10667097 0.72 HIF1A (0.49) HIF1AALDH1A1TAAR1TDP1KDM4E
SCHEMBL10670005 0.71 ADRB1 (0.39) HIF1AKDM4EHTR1ABLMCYP2C9
SCHEMBL10671463 0.70 ALDH1A1 (0.36) HIF1AALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL10663271 0.69 ALDH1A1 (0.49) ALDH1A1TDP1KDM4ESMN1; SMN2ADRB2
SCHEMBL6458210 0.65 HIF1A (0.61) HIF1AALDH1A1TAAR1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4721717-A α-(aminoalkylaminomethyl)phenylmethanols, composition containing them, and use thereof to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-01-26 US disclosed