SCHEMBL10685641

SCHEMBL10685641

COC(=O)CCSc1scnc1C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.39
GSTP1 P09211 1/20 0.34
GSTM2 P28161 1/20 0.34
CCNB2 O95067 1/20 0.34
CCNE2 O96020 1/20 0.34
CDK1 P06493 1/20 0.34
CDK4 P11802 1/20 0.34
CCNB1 P14635 1/20 0.34
CCND1 P24385 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CCNB3 Q8WWL7 1/20 0.34
CXCR1 P25024 1/20 0.33
CXCR2 P25025 1/20 0.33
ALDH1A1 P00352 4/20 0.32
LMNA P02545 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852499 0.83 KMT2A (0.40) PTGS1GSTP1GSTM2CXCR1CXCR2
SCHEMBL9748843 0.81 PTGS1 (0.38) PTGS1GSTP1GSTM2CCNB2CCNE2
SCHEMBL10688854 0.74 HSD17B10 (0.43) ALDH1A1KMT2AMEN1HSD17B10KDM4E
SCHEMBL9748003 0.73 PTGS1 (0.36) PTGS1GSTP1GSTM2CXCR1CXCR2
SCHEMBL9852546 0.73 PTGS1 (0.36) PTGS1GSTP1GSTM2CXCR1CXCR2
SCHEMBL10690505 0.71 NPSR1 (0.38) ALDH1A1LMNAKMT2AMEN1RAB9A
SCHEMBL9627261 0.70 KDM4E (0.43) ALDH1A1LMNAKMT2AMEN1RAB9A
SCHEMBL15737155 0.69 KMT2A (0.43) PTGS1GSTP1GSTM2CXCR1CXCR2
SCHEMBL22589563 0.68 GRM6 (0.38) ALDH1A1LMNACYP1A2CYP2C9CYP2C19
SCHEMBL16311074 0.68 ALDH1A1 (0.36) ALDH1A1LMNACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4762848-A IMMUNE SYSTEM STIMULANTS, CYTOSTATIC AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1988-08-09 US disclosed