SCHEMBL9748843

SCHEMBL9748843

COC(=O)CCSc1scnc1OC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.38
CCNE2 O96020 2/20 0.35
CCNE1 P24864 2/20 0.35
CDK2 P24941 2/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCNB1 P14635 1/20 0.35
CCND1 P24385 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
CXCR1 P25024 1/20 0.32
CXCR2 P25025 1/20 0.32
VCAM1 P19320 1/20 0.32
GSTP1 P09211 1/20 0.31
GSTM2 P28161 1/20 0.31
ELANE P08246 1/20 0.31
HPGD P15428 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852546 0.89 PTGS1 (0.36) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL9748003 0.84 PTGS1 (0.36) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL10685641 0.81 PTGS1 (0.39) PTGS1CCNE2CCNE1CDK2CCNB2
SCHEMBL9749147 0.76 MAPK1 (0.40) HPGDALDH1A1MAPTKMT2AHSD17B10
SCHEMBL9852499 0.73 KMT2A (0.40) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL9748133 0.72 HSD17B10 (0.32) HPGDALDH1A1MAPTHSD17B10
SCHEMBL15737155 0.65 KMT2A (0.43) PTGS1CXCR1CXCR2GSTP1GSTM2
SCHEMBL12292 0.64 CCNE1 (0.59) PTGS1CCNE2CCNE1CDK2CCNB2
SCHEMBL6760169 0.64 KDM4E (0.40) PTGS1LMNAHTTKMT2A
SCHEMBL9627350 0.63 PTGS1 (0.40) PTGS1CXCR1CXCR2GSTP1GSTM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0194572-B1 HETEROCYCLIC SULFIDES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-01-02 EP disclosed