SCHEMBL10690528

SCHEMBL10690528

OCC1CN(CCN2CCCC2)CCc2c1[nH]c1ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.56
ADRA1D P25100 2/20 0.51
ADRA1A P35348 2/20 0.51
ADRA1B P35368 2/20 0.51
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
ESR1 P03372 2/20 0.48
PGR P06401 1/20 0.48
BRD3 Q15059 1/20 0.44
ABCB1 P08183 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
LMNA P02545 1/20 0.43
STAT3 P40763 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
PDE5A O76074 2/20 0.42
PRKCB P05771 1/20 0.42
CYP1A1 P04798 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10686642 0.99 SIGMAR1 (0.55) SIGMAR1ADRA1DADRA1AADRA1BCYP2D6
SCHEMBL10690885 0.91 LMNA (0.52) SIGMAR1ADRA1DADRA1AADRA1BCYP2D6
SCHEMBL10685213 0.88 ADRA1D (0.51) SIGMAR1ADRA1DADRA1AADRA1BCYP2D6
SCHEMBL10686306 0.85 ADRA1D (0.53) SIGMAR1ADRA1DADRA1AADRA1BESR1
SCHEMBL10681421 0.85 ADRA1D (0.48) SIGMAR1ADRA1DADRA1AADRA1BESR1
SCHEMBL10682913 0.83 ACHE (0.54) SIGMAR1ADRA1DADRA1AADRA1BESR1
SCHEMBL10687988 0.83 ADRA1D (0.46) SIGMAR1ADRA1DADRA1AADRA1BESR1
SCHEMBL10688707 0.83 ADRA1D (0.56) SIGMAR1ADRA1DADRA1AADRA1BCYP2D6
SCHEMBL10690521 0.79 ADRA1D (0.49) SIGMAR1ADRA1DADRA1AADRA1BESR1
SCHEMBL10686635 0.78 ADRA1D (0.48) SIGMAR1ADRA1DADRA1AADRA1BESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4719208-A 1,2,3,4,5,6-hexahydroazepino(4,5-B)indole derivatives, their preparation, intermediate compounds, and their application in therapeutics OMNICHEM SOCIETE ANONYME (BE) 1988-01-12 US disclosed