SCHEMBL10690885

SCHEMBL10690885

OCC1CN(CCN2CCOCC2)CCc2c1[nH]c1ccccc21

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
STAT3 P40763 1/20 0.52
ADRA1D P25100 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
SIGMAR1 Q99720 2/20 0.47
ESR1 P03372 2/20 0.47
PGR P06401 1/20 0.47
CYP2D6 P10635 3/20 0.46
KDM4E B2RXH2 1/20 0.44
ABCB1 P08183 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10690528 0.91 SIGMAR1 (0.56) LMNASTAT3ADRA1DADRA1AADRA1B
SCHEMBL10686642 0.90 SIGMAR1 (0.55) LMNASTAT3ADRA1DADRA1AADRA1B
SCHEMBL10685213 0.86 ADRA1D (0.51) ADRA1DADRA1AADRA1BSIGMAR1ESR1
SCHEMBL10686306 0.83 ADRA1D (0.53) ADRA1DADRA1AADRA1BSIGMAR1ESR1
SCHEMBL10681421 0.83 ADRA1D (0.48) ADRA1DADRA1AADRA1BSIGMAR1ESR1
SCHEMBL10682913 0.81 ACHE (0.54) LMNAADRA1DADRA1AADRA1BSIGMAR1
SCHEMBL10690877 0.81 KDM4E (0.48) LMNASTAT3ADRA1DADRA1AADRA1B
SCHEMBL10687988 0.81 ADRA1D (0.46) ADRA1DADRA1AADRA1BSIGMAR1ESR1
SCHEMBL10688707 0.81 ADRA1D (0.56) ADRA1DADRA1AADRA1BSIGMAR1ESR1
SCHEMBL10682960 0.74 DRD2 (0.48) LMNAADRA1DADRA1AADRA1BESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4719208-A 1,2,3,4,5,6-hexahydroazepino(4,5-B)indole derivatives, their preparation, intermediate compounds, and their application in therapeutics OMNICHEM SOCIETE ANONYME (BE) 1988-01-12 US disclosed
EP-0203902-A2 1,2,3,4,5,6-Hexahydro-azepino[4,5-b] indole derivatives, their preparation, intermediate compounds and their therapeutical use OMNICHEM Société anonyme (BE) 1986-12-03 EP disclosed