SCHEMBL10690584

SCHEMBL10690584

CN1C(=O)C(C)(c2ccccc2OCCCCBr)Cc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
POLB P06746 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DRD2 P14416 4/20 0.35
HTT P42858 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
NQO1 P15559 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
HTR1A P08908 1/20 0.32
HTR2A P28223 1/20 0.32
MAPK1 P28482 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694109 0.85 POLB (0.35) ALDH1A1POLBHSD17B10DRD2HTT
SCHEMBL10693548 0.84 RAD52 (0.35) ALDH1A1POLBHSD17B10DRD2HTT
SCHEMBL10696619 0.83 RAD52 (0.34) ALDH1A1POLBHSD17B10DRD2HTT
SCHEMBL10694576 0.82 POLB (0.33) ALDH1A1POLBHSD17B10DRD2HTT
SCHEMBL10689170 0.81 ADRA1A (0.40) ALDH1A1DRD2HTTMAPTADRA1D
SCHEMBL10692777 0.81 OPRL1 (0.35) ALDH1A1POLBHSD17B10DRD2MAPT
SCHEMBL10694665 0.81 RAD52 (0.36) ALDH1A1POLBHSD17B10DRD2HTT
SCHEMBL10691826 0.78 HTR2A (0.43) ALDH1A1POLBDRD2HTTL3MBTL1
Hydrochloric Acid SCHEMBL10695977 0.76 DRD2 (0.42) ALDH1A1DRD2ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL10693968 0.76 SMPD1 (0.52) DRD2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed