SCHEMBL10694576

SCHEMBL10694576

CN1C(=O)C(Cc2ccccc2)(c2ccccc2OCCCCBr)Cc2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.33
HSD17B10 Q99714 1/20 0.33
DRD2 P14416 3/20 0.33
HTT P42858 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
HCRTR1 O43613 1/20 0.32
LMNA P02545 1/20 0.32
ALDH1A1 P00352 3/20 0.31
BACE1 P56817 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
ITGB2 P05107 1/20 0.31
ICAM1 P05362 1/20 0.31
ITGAL P20701 1/20 0.31
HTR7 P34969 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
BCHE P06276 1/20 0.31
ADRA1D P25100 2/20 0.31
ADRA1A P35348 2/20 0.31
ADRA1B P35368 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694109 0.89 POLB (0.35) POLBHSD17B10DRD2HTTKDM4E
SCHEMBL10692777 0.84 OPRL1 (0.35) POLBHSD17B10DRD2MAPTLMNA
SCHEMBL10695992 0.84 SCN9A (0.39) KDM4EMAPTHCRTR1LMNAALDH1A1
SCHEMBL10690584 0.82 ALDH1A1 (0.36) POLBHSD17B10DRD2HTTMAPT
SCHEMBL10759482 0.80 SLC6A3 (0.42) DRD2HTTKDM4EMAPTLMNA
SCHEMBL10370705 0.80 ALDH1A1 (0.36) KDM4EMAPTHCRTR1LMNAALDH1A1
SCHEMBL10693548 0.80 RAD52 (0.35) POLBHSD17B10DRD2HTTMAPT
SCHEMBL10763371 0.80 HTR1A (0.42) DRD2KDM4EALDH1A1TDP1
Hydrochloric Acid SCHEMBL10692827 0.80 SLC6A3 (0.42) DRD2HTTKDM4EMAPTLMNA
SCHEMBL10757925 0.80 SMPD1 (0.50) KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed