SCHEMBL10695791

SCHEMBL10695791

C=CCc1nccc(C(N)=O)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.34
TSHR P16473 1/20 0.34
MC4R P32245 1/20 0.34
ADRA1A P35348 1/20 0.34
MC3R P41968 1/20 0.34
KDM4E B2RXH2 2/20 0.33
KDM5A P29375 1/20 0.33
JMJD1C Q15652 1/20 0.33
KDM3A Q9Y4C1 1/20 0.33
PARP1 P09874 1/20 0.33
PIM1 P11309 1/20 0.33
LMNA P02545 1/20 0.32
KMT2A Q03164 2/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
MEN1 O00255 1/20 0.31
PKM P14618 1/20 0.31
HPGD P15428 1/20 0.31
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826624 0.77 ADORA3 (0.37) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL13729259 0.76 SORD (0.40) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL13728021 0.75 KDM4E (0.39) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL8918530 0.74
SCHEMBL8918540 0.74
SCHEMBL6305112 0.73 NNMT (0.39) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL29519619 0.73 NR3C2 (0.35) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL1257943 0.73 IMPDH2 (0.37)
SCHEMBL532603 0.73 XDH (0.34) KDM4EKMT2AMEN1HPGD
SCHEMBL163636 0.72 ADORA3 (0.42) ADORA3TSHRMC4RADRA1AMC3R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4794182-A 2-Alkyl-4-amino-5-aminomethylpyrimidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-12-27 US disclosed