SCHEMBL10697202

SCHEMBL10697202

CCN1C(=O)C(C)(C)c2cc3c(cc21)NC(c1ccc(SC)cc1OC)N3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
HSD11B1 P28845 2/20 0.36
AURKA O14965 2/20 0.33
AURKB Q96GD4 2/20 0.33
HPGD P15428 6/20 0.32
POLB P06746 2/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 3/20 0.32
KDM4E B2RXH2 2/20 0.32
HSD17B10 Q99714 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA1A P35348 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CHEK1 O14757 1/20 0.30
SRC P12931 1/20 0.30
CDK2 P24941 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10697456 0.83 MEN1 (0.40) ALDH1A1L3MBTL1AURKAAURKBHPGD
SCHEMBL10373869 0.78 PGR (0.39) ALDH1A1L3MBTL1HSD11B1HPGDPOLB
SCHEMBL10701198 0.77 TNKS2 (0.44) ALDH1A1L3MBTL1HSD11B1AURKAAURKB
SCHEMBL10696440 0.76 MEN1 (0.40) ALDH1A1L3MBTL1AURKAAURKBHPGD
SCHEMBL10696613 0.74 AURKA (0.40) ALDH1A1L3MBTL1AURKAAURKBHPGD
SCHEMBL10697356 0.73 MEN1 (0.40) ALDH1A1HPGDKDM4EHSD17B10MEN1
SCHEMBL10698519 0.72 CNR1 (0.41) ALDH1A1AURKAAURKBLMNAMEN1
SCHEMBL10698153 0.72 AURKA (0.38) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10700532 0.72 AURKA (0.43) ALDH1A1AURKAAURKBLMNAMEN1
SCHEMBL10699508 0.72 AURKA (0.39) AURKAAURKBCHEK1SRCCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed