SCHEMBL10700249

SCHEMBL10700249

O=c1c2ccccc2c(Cc2ccc(F)cc2)nn1CCN(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 8/20 0.57
HRH1 P35367 8/20 0.57
ADRA1B P35368 8/20 0.57
TSHR P16473 1/20 0.54
HRH3 Q9Y5N1 4/20 0.53
GLA P06280 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
KCNH2 Q12809 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10482471 0.89 ADRA1A (0.61) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL10700164 0.86 ADRA1A (0.55) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL10700300 0.80 ADRA1A (0.55) ADRA1AHRH1ADRA1BTSHRHRH3
Talastine SCHEMBL29350005 0.79 ADRA1A (0.81) ADRA1AHRH1ADRA1BTSHRHRH3
Talastine SCHEMBL30502 0.79 ADRA1A (0.81) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL10698694 0.79 ADRA1A (0.62) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL10700979 0.78 HRH1 (0.65) ADRA1AHRH1ADRA1BHRH3KCNH2
Talastine SCHEMBL1650995 0.77 ADRA1A (0.78) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL7884616 0.76 TSHR (0.52) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL7894969 0.74 TSHR (0.66) ADRA1AHRH1ADRA1BTSHRGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289881-A2 2-Aminoalkyl-4-benzyl-1-(2H)-phthalazinone derivatives ASTA Medica Aktiengesellschaft (DE) 1988-11-09 EP disclosed