SCHEMBL10698694

SCHEMBL10698694

CNCCn1nc(Cc2ccc(F)cc2)c2ccccc2c1=O

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 10/20 0.62
HRH1 P35367 10/20 0.62
ADRA1B P35368 10/20 0.62
HRH3 Q9Y5N1 5/20 0.54
TSHR P16473 1/20 0.52
USP2 O75604 1/20 0.49
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10700300 0.86 ADRA1A (0.55) ADRA1AHRH1ADRA1BHRH3TSHR
SCHEMBL13890824 0.80 HRH1 (0.72) ADRA1AHRH1ADRA1BHRH3TSHR
SCHEMBL10482471 0.79 ADRA1A (0.61) ADRA1AHRH1ADRA1BHRH3TSHR
SCHEMBL10700249 0.79 ADRA1A (0.57) ADRA1AHRH1ADRA1BHRH3TSHR
SCHEMBL10700979 0.78 HRH1 (0.65) ADRA1AHRH1ADRA1BHRH3KCNH2
SCHEMBL10700164 0.77 ADRA1A (0.55) ADRA1AHRH1ADRA1BHRH3TSHR
SCHEMBL7894969 0.75 TSHR (0.66) ADRA1AHRH1ADRA1BTSHRUSP2
Bromide SCHEMBL9690249 0.74 RAB9A (0.59) TSHRLMNASMN1; SMN2
SCHEMBL16363659 0.74 TSHR (0.64) ADRA1AHRH1ADRA1BHRH3TSHR
Talastine SCHEMBL30502 0.73 ADRA1A (0.81) ADRA1AHRH1ADRA1BHRH3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289881-A2 2-Aminoalkyl-4-benzyl-1-(2H)-phthalazinone derivatives ASTA Medica Aktiengesellschaft (DE) 1988-11-09 EP disclosed