SCHEMBL10700300

SCHEMBL10700300

O=c1c2ccccc2c(Cc2ccc(F)cc2)nn1CCNCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 7/20 0.55
HRH1 P35367 7/20 0.55
ADRA1B P35368 7/20 0.55
TSHR P16473 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.48
USP2 O75604 1/20 0.48
LMNA P02545 1/20 0.48
HRH3 Q9Y5N1 4/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
GLA P06280 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698694 0.86 ADRA1A (0.62) ADRA1AHRH1ADRA1BTSHRSMN1; SMN2
SCHEMBL7894969 0.81 TSHR (0.66) ADRA1AHRH1ADRA1BTSHRSMN1; SMN2
SCHEMBL10700249 0.80 ADRA1A (0.57) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL10482471 0.78 ADRA1A (0.61) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL10700164 0.75 ADRA1A (0.55) ADRA1AHRH1ADRA1BTSHRSMN1; SMN2
SCHEMBL16363659 0.73 TSHR (0.64) ADRA1AHRH1ADRA1BTSHRHRH3
SCHEMBL7885318 0.72 TSHR (0.76) TSHRLMNACYP1A2CYP3A4CYP2C9
SCHEMBL12877772 0.72 TSHR (0.71) ADRA1AHRH1ADRA1BTSHRHRH3
Talastine SCHEMBL29350005 0.72 ADRA1A (0.81) ADRA1AHRH1ADRA1BTSHRHRH3
Talastine SCHEMBL30502 0.72 ADRA1A (0.81) ADRA1AHRH1ADRA1BTSHRHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289881-A2 2-Aminoalkyl-4-benzyl-1-(2H)-phthalazinone derivatives ASTA Medica Aktiengesellschaft (DE) 1988-11-09 EP disclosed