SCHEMBL10700609

SCHEMBL10700609

CCCCCN1C(=O)C(C)(C)c2cc3c(cc21)NC(c1cnccn1)N3

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.32
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32
CYP19A1 P11511 11/20 0.31
KCNA5 P22460 1/20 0.31
KCNJ5 P48544 1/20 0.31
KCNJ3 P48549 1/20 0.31
CNR2 P34972 2/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10697407 0.89 AURKA (0.40) AURKAAURKBKCNA5KCNJ5KCNJ3
SCHEMBL10695491 0.84 MAPT (0.42) SCN9ACNR2
SCHEMBL10693698 0.83 KDM4E (0.40) SCN9ACYP19A1CNR2
SCHEMBL10695292 0.82 PDE4A (0.38) ADORA2A
SCHEMBL10696477 0.80 KDM4E (0.42) KCNA5KCNJ5KCNJ3
SCHEMBL10696397 0.80 ALDH1A1 (0.40) CYP19A1
SCHEMBL10696318 0.78 KDM4E (0.41) KCNA5KCNJ5KCNJ3
SCHEMBL10696042 0.77 ALDH1A1 (0.39) AURKAAURKBCYP19A1KCNA5KCNJ5
SCHEMBL10695201 0.75 SCN9A (0.35) SCN9ACNR2ADORA2B
SCHEMBL10695114 0.75 SCN9A (0.37) SCN9ACNR2ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed