SCHEMBL10696397

SCHEMBL10696397

CCCCN1C(=O)C(C)(C)c2cc3c(cc21)NC(c1ccncc1)N3

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP19A1 P11511 14/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
ALOX12 P18054 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10693698 0.97 KDM4E (0.40) ALDH1A1KDM4EHSD17B10CYP19A1
SCHEMBL10696042 0.93 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10CYP19A1HPGD
SCHEMBL10696613 0.90 AURKA (0.40) ALDH1A1KDM4EHSD17B10CYP19A1KMT2A
SCHEMBL10698603 0.87 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL10696477 0.87 KDM4E (0.42) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL10695087 0.87 TNKS2 (0.44) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL10698037 0.86 ALDH1A1 (0.38) ALDH1A1KDM4EHSD17B10MAPTTDP1
SCHEMBL10695491 0.84 MAPT (0.42) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL10694215 0.82 ELANE (0.46) ALDH1A1KDM4EHSD17B10MAPTTDP1
SCHEMBL10695498 0.82 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed