SCHEMBL107330

SCHEMBL107330

Clc1cnc2n1CCNC2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.36
HTR2C P28335 4/20 0.36
WNT1 P04628 4/20 0.36
GSK3B P49841 4/20 0.36
DYRK1A Q13627 4/20 0.36
ADRB2 P07550 1/20 0.35
P2RX7 Q99572 1/20 0.35
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL708722 0.77 CHRNB2 (0.36) HTR2AHTR2CWNT1GSK3BDYRK1A
SCHEMBL928582 0.77 HTR2A (0.36) HTR2AHTR2CWNT1GSK3BDYRK1A
SCHEMBL17687467 0.77 GSK3B (0.36) HTR2AHTR2CWNT1GSK3BDYRK1A
Hydrochloric Acid SCHEMBL930044 0.76 HTR2A (0.36) HTR2AHTR2CWNT1GSK3BDYRK1A
SCHEMBL24024593 0.73 GSK3B (0.34) WNT1GSK3BDYRK1A
SCHEMBL10183608 0.73 GSK3B (0.34) WNT1GSK3BDYRK1A
SCHEMBL17788669 0.73 GSK3B (0.35) WNT1GSK3BDYRK1ACHRNB2CHRNA4
SCHEMBL13193521 0.73 CPB2 (0.39) HTR2CWNT1GSK3BDYRK1A
SCHEMBL31509704 0.73 MGLL (0.39) HTR2AHTR2CWNT1GSK3BDYRK1A
SCHEMBL2556005 0.73 GSK3B (0.36) HTR2AHTR2CWNT1GSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119661811-A Latent accelerator based on anhydride-tertiary amine dynamic ion pair, preparation method and application thereof 江南大学 2025-03-21 CN claimed
CN-119661811-A Latent accelerator based on anhydride-tertiary amine dynamic ion pair, preparation method and application thereof 江南大学 2025-03-21 CN disclosed
EP-2424867-B1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LTD (GB) 2013-09-18 EP disclosed
EP-2424867-B1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LTD (GB) 2013-09-18 EP disclosed
US-8513248-B2 5,6,7,8-tetrahydroimidazo[1,2-A]pyrazine derivatives as P2X7 modulators GLAXO GROUP LIMITED (GB) 2013-08-20 US disclosed
US-8513248-B2 5,6,7,8-tetrahydroimidazo[1,2-A]pyrazine derivatives as P2X7 modulators GLAXO GROUP LIMITED (GB) 2013-08-20 US disclosed
US-8513248-B2 5,6,7,8-tetrahydroimidazo[1,2-A]pyrazine derivatives as P2X7 modulators GLAXO GROUP LIMITED (GB) 2013-08-20 US disclosed
US-20120172366-A1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2012-07-05 US disclosed
US-20120172366-A1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2012-07-05 US disclosed
US-20120172366-A1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2012-07-05 US disclosed
EP-2424867-A1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS Glaxo Group Limited (GB) 2012-03-07 EP disclosed
WO-2010125101-A1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2010-11-04 WO disclosed
WO-2010125101-A1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2010-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120172366-A1 5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRAZINE DERIVATIVES AS P2X7 MODULATORS P2RX7, P2RX6, P2RX3 HTR2A 279/4885HTR2C 182/4885WNT1 574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.