SCHEMBL10745926

SCHEMBL10745926

COc1cc2c(cc1OC)n1c(=O)[nH]nc1c(=O)n2C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.40
S100B P04271 1/20 0.40
ADORA1 P30542 1/20 0.34
CHEK1 O14757 2/20 0.34
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 3/20 0.33
RET P07949 2/20 0.33
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
GLA P06280 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10742951 0.83 KDM4E (0.42) CHEK1ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL10743293 0.82 MTNR1B (0.42) ADORA1CHEK1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL11069723 0.81 LMNA (0.44) ADORA1CHEK1ALDH1A1KDM4ERET
SCHEMBL10744610 0.77 PARP10 (0.49) CHEK1ALDH1A1KDM4EPDE3BPDE3A
SCHEMBL10746913 0.77 PARP10 (0.49) CHEK1ALDH1A1KDM4EPDE3BPDE3A
SCHEMBL10747539 0.75 ADORA3 (0.50) ADORA1CHEK1RETSMN1; SMN2PDE3B
SCHEMBL10744197 0.75 KDM4E (0.41) ALDH1A1KDM4EHPGDSMN1; SMN2GLA
SCHEMBL10745104 0.72 KDM4E (0.40) ADORA1ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL10745368 0.72 CYP1A2 (0.40) CYP2C9ALDH1A1KMT2ACYP1A2
Potassium Ion SCHEMBL10743069 0.70 ALDH1A1 (0.37) CHEK1ALDH1A1KDM4ESMN1; SMN2GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4668678-A ANTIALLERGENS USV PHARMACEUTICAL CORPORATION (US) 1987-05-26 US disclosed
US-4507300-A Pyridotriazolopyrazine-diones for treating allergy USV PHARMACEUTICAL CORPORATION (US) 1985-03-26 US disclosed
US-4400382-A Thiazoloquinoxalin-1,4-diones for treating allergy USV PHARMACEUTICAL CORPORATION (US) 1983-08-23 US disclosed
EP-0039920-A2 Triazaloquinoxalin-1,4-diones USV PHARMACEUTICAL CORPORATION (US) 1981-11-18 EP disclosed