SCHEMBL11017363

SCHEMBL11017363

CCCSc1ccc(-c2nc3ccc(C#N)cc3[nH]2)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.50
CYP1A2 P05177 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
HPGD P15428 1/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNH2 Q12809 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CYP2E1 P05181 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2B6 P20813 1/20 0.45
CYP2C19 P33261 1/20 0.45
PKN1 Q16512 1/20 0.44
PKN2 Q16513 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11017329 0.92 AR (0.50) ARCYP1A2MEN1LMNATP53
SCHEMBL11018943 0.92 AMY1A (0.47) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL11019300 0.86 PKN1 (0.48) PKN1PKN2AMY1ACFBCHEK2
SCHEMBL10762222 0.83 AMY1A (0.41) ARCYP1A2MEN1HPGDKMT2A
SCHEMBL11016890 0.80 CHEK2 (0.63) CYP1A2MEN1LMNATP53HPGD
SCHEMBL11021674 0.79 METAP2 (0.46) LMNATP53HPGDKCNH2SMN1; SMN2
SCHEMBL11018186 0.78 CYP3A4 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11018077 0.78 CYP2C9 (0.54) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11021164 0.78 PKN1 (0.42) PKN1PKN2AMY1ACFBCHEK2
SCHEMBL7271872 0.78 PDE5A (0.48) ARCYP1A2MEN1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed