SCHEMBL11018943

SCHEMBL11018943

CCSc1ccc(-c2nc3ccc(C#N)cc3[nH]2)c(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 7/20 0.47
PKN1 Q16512 1/20 0.46
PKN2 Q16513 1/20 0.46
CFB P00751 7/20 0.44
CHEK2 O96017 1/20 0.43
METAP2 P50579 1/20 0.43
METAP1 P53582 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
CYP2C19 P33261 1/20 0.43
F7 P08709 1/20 0.42
ALOX5 P09917 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11017363 0.92 AR (0.50) AMY1APKN1PKN2CFBCHEK2
SCHEMBL10762222 0.92 AMY1A (0.41) AMY1APKN1PKN2CFBCYP1A2
SCHEMBL11019300 0.88 PKN1 (0.48) AMY1APKN1PKN2CFBCHEK2
SCHEMBL11017329 0.83 AR (0.50) AMY1APKN1PKN2CFBCYP1A2
SCHEMBL11021674 0.81 METAP2 (0.46) PKN1PKN2CFBCHEK2METAP2
SCHEMBL11017902 0.80 CHEK2 (0.53) AMY1ACHEK2
SCHEMBL11018186 0.80 CYP3A4 (0.48) PKN1PKN2CFBCYP1A2CYP3A4
SCHEMBL11016463 0.79 CHEK2 (0.66) CHEK2
SCHEMBL11018211 0.79 CHEK2 (0.47) AMY1APKN1PKN2CFBCHEK2
SCHEMBL11018557 0.79 PKN1 (0.44) AMY1APKN1PKN2CFBCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed