SCHEMBL10846355

SCHEMBL10846355

CC1CN(c2cccc(Cl)n2)N=C1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 3/20 0.44
HTR3B O95264 3/20 0.44
HTR3A P46098 3/20 0.44
HTR3D Q70Z44 3/20 0.44
HTR3C Q8WXA8 3/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
TSHR P16473 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
ALOX5 P09917 2/20 0.44
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
CHRM4 P08173 2/20 0.34
PTPN11 Q06124 2/20 0.33
ROCK1 Q13464 1/20 0.33
GRM4 Q14833 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10850373 0.83 ALOX5 (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL908132 0.76 HSD11B1 (0.40) ALOX15KDM4EROCK1HSD11B1
SCHEMBL11242467 0.74 ABL1 (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL908243 0.73 DHFR (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL908503 0.72 ROCK1 (0.40) HTR3AALDH1A1PTPN11ROCK1
SCHEMBL7721894 0.71 BRD4 (0.39) KMT2AMEN1ALDH1A1
SCHEMBL10850532 0.70 HTR3E (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL10846913 0.70 HTR3E (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9005356 0.69 KMT2A (0.50) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7382691 0.67 HTR3E (0.70) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4622401-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS AMERICAN CYANAMID COMPANY (US) 1986-11-11 US disclosed
EP-0070376-A1 Heterocyclic substituted-amino-pyrazolines AMERICAN CYANAMID COMPANY (US) 1983-01-26 EP disclosed
US-4347251-A ANTIINFLAMMATORY, ANALGESICS, BACTERICIDES, FUNGICIDES AMERICAN CYANAMID COMPANY (US) 1982-08-31 US disclosed