SCHEMBL10872018

SCHEMBL10872018

C[C@@H]1CN(C[C@@H]2C[C@H]2c2ccc([Si](C)(C)C)cc2)C[C@H](C)O1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.38
DRD4 P21917 10/20 0.38
KDM1A O60341 1/20 0.38
KDM4E B2RXH2 2/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
OPRM1 P35372 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP2A13 Q16696 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691883 0.82 SIGMAR1 (0.52) DRD2DRD4KDM1AKDM4EHTT
SCHEMBL9820772 0.70 NPC1 (0.44)
SCHEMBL10685814 0.69 SIGMAR1 (0.39) KDM1AKDM4EHTTLMNAGAA
SCHEMBL10694936 0.68 SIGMAR1 (0.40) KDM4EHTTLMNAGAATDP1
SCHEMBL10682744 0.68 SIGMAR1 (0.38) KDM1AKDM4EHTTLMNAGAA
SCHEMBL5802152 0.67 HRH3 (0.44) KDM4E
SCHEMBL10929087 0.66 SIGMAR1 (0.69) KDM4EHTTLMNAGAA
SCHEMBL10929081 0.66 SIGMAR1 (0.69) KDM4EHTTLMNAGAA
SCHEMBL9821040 0.61 FFAR1 (0.55)
SCHEMBL9821161 0.61 ALDH1A1 (0.42) HTTLMNAGAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188887-A1 Tertiary amine compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-07-30 EP disclosed