SCHEMBL10909110

SCHEMBL10909110

O=C(Nc1ccc(C(=O)Nc2c(O)ccc3ccc(S(=O)(=O)O)cc23)cc1)C(=O)Nc1ccc(C(=O)Nc2c(O)ccc3ccc(S(=O)(=O)O)cc23)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTDSP1 Q9GZU7 2/20 0.50
CASP6 P55212 1/20 0.50
CA1 P00915 4/20 0.46
CA2 P00918 4/20 0.46
ENPP2 Q13822 2/20 0.44
TIMP3 P35625 2/20 0.44
NT5E P21589 1/20 0.43
PRMT1 Q99873 1/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
APEX1 P27695 1/20 0.42
TOP1 P11387 1/20 0.41
MEN1 O00255 6/20 0.41
KMT2A Q03164 6/20 0.41
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PSMD14 O00487 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11338837 0.93 TIMP3 (0.53) CTDSP1CASP6CA1CA2ENPP2
SCHEMBL10907702 0.92 CASP6 (0.55) CTDSP1CASP6CA1CA2ENPP2
SCHEMBL10909529 0.87 KMT2A (0.46) CTDSP1CASP6TIMP3NT5EPRMT1
SCHEMBL11440941 0.86 CASP6 (0.60) CTDSP1CASP6CA1CA2ENPP2
SCHEMBL11350531 0.84 PRMT1 (0.57) CTDSP1CASP6CA1CA2ENPP2
SCHEMBL11431481 0.83 RAB9A (0.56) CTDSP1CASP6CA1CA2CA9
SCHEMBL10905197 0.83 CASP6 (0.59) CTDSP1CASP6CA1CA2ENPP2
SCHEMBL10909096 0.83 TIMP3 (0.50) CTDSP1CASP6CA1CA2ENPP2
SCHEMBL10909449 0.83 NT5E (0.42) CTDSP1CASP6CA2NT5EPRMT1
SCHEMBL10908164 0.81 TIMP3 (0.51) CTDSP1CASP6CA1CA2TIMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4599204-A Oxalylamides useful as dental antiplaque agents and inhibitors of connective tissue destruction AMERICAN CYANAMID COMPANY (US) 1986-07-08 US disclosed