SCHEMBL10945238

SCHEMBL10945238

COC(=O)CNC(=O)[C@@H](C)N(C(=O)OC(C)(C)C)C(=O)[C@@H](N)Cc1ccc(OCc2c(Cl)cccc2Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 15/20 0.41
ITGB1 P05556 4/20 0.41
MAOB P27338 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10947130 1.00 ITGA4 (0.41) ITGA4ITGB1MAOB
SCHEMBL10939289 0.93 ITGA4 (0.41) ITGA4ITGB1MAOB
SCHEMBL11349836 0.82 LTA4H (0.45) MAOB
SCHEMBL11357211 0.78 PSMB10 (0.44)
SCHEMBL10939294 0.77 OPRD1 (0.43) ITGA4ITGB1
SCHEMBL11525876 0.76 PSMB1 (0.50)
SCHEMBL5719618 0.76 ITGA4 (0.48) ITGA4ITGB1
SCHEMBL5719732 0.76 ITGA4 (0.48) ITGA4ITGB1
SCHEMBL10945240 0.76 REN (0.53) ITGA4ITGB1
SCHEMBL11349851 0.75 LTA4H (0.48) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4534897-A Piperazinone, piperazine, 1,4-diazepin-2-one and 1,4-diazepine intermediate compounds THE UPJOHN COMPANY (US) 1985-08-13 US disclosed
US-4251438-A ANALGESICS, PSYCHOTHERAPEUTIC AGENTS THE UPJOHN COMPANY (US) 1981-02-17 US disclosed