SCHEMBL1094563

SCHEMBL1094563

O=S(=O)(Nc1ncns1)c1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 13/20 0.55
SLC40A1 Q9NP59 3/20 0.50
GLO1 Q04760 1/20 0.50
SCN5A Q14524 3/20 0.47
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
SCN1A P35498 1/20 0.46
SCN8A Q9UQD0 1/20 0.46
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1093900 0.83 SCN9A (0.59) SCN9ASCN5ASCN1ASCN8A
SCHEMBL3476554 0.78 ALDH1A1 (0.60) SLC40A1GLO1KMT2A
SCHEMBL1093897 0.75 SCN9A (0.59) SCN9ASCN5A
SCHEMBL29835215 0.75 SCN9A (0.59) SCN9ASCN5A
SCHEMBL18885650 0.74 SCN9A (0.56) SCN9ASCN5A
SCHEMBL1576706 0.74 CA12 (0.51) SCN9ASCN5ASCN1ASCN8A
SCHEMBL1094451 0.72 SCN9A (0.62) SCN9ASLC40A1GLO1SCN5A
SCHEMBL28886252 0.72 SCN9A (0.52) SCN9ASCN5ASCN1ASCN8A
SCHEMBL6292016 0.72 SLC40A1 (0.55) SLC40A1GLO1KEAP1NFE2L2KMT2A
SCHEMBL1093538 0.72 SLC40A1 (0.48) SLC40A1GLO1KEAP1NFE2L2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8907101-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2014-12-09 US disclosed
US-20130338111-A1 Sulfonamide Derivatives ICAGEN, INC. (US) 2013-12-19 US disclosed
US-20120149679-A1 Sulfonamide Derivatives ICAGEN, INC. 2012-06-14 US disclosed
US-8153814-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2012-04-10 US disclosed
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197655-A1 SULFONAMIDE DERIVATIVES SULT2A1, SULT1A1, TPST2 SCN9A 73/4885SLC40A1 3958/4885GLO1 2222/4885
US-20130338111-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 SCN9A 73/4885SLC40A1 3958/4885GLO1 2222/4885
US-20120149679-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 SCN9A 73/4885SLC40A1 3958/4885GLO1 2222/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.