SCHEMBL11022178

SCHEMBL11022178

CCOC(=O)c1c(CC)[nH]c2cc(C#N)c(F)cc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
MAPT P10636 6/20 0.40
ALDH1A1 P00352 5/20 0.40
KMT2A Q03164 5/20 0.40
MEN1 O00255 3/20 0.40
RXFP1 Q9HBX9 1/20 0.40
STAT3 P40763 1/20 0.39
KDM4E B2RXH2 6/20 0.39
GLA P06280 1/20 0.39
ATM Q13315 1/20 0.39
POLB P06746 3/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
PKM P14618 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB2 P47870 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7113113 0.76 ALDH1A1 (0.45) NPC1MAPTALDH1A1KMT2AMEN1
SCHEMBL4961457 0.73 GABRA1 (0.54) MAPTALDH1A1KMT2AMEN1KDM4E
SCHEMBL17769795 0.72 MAPT (0.46) NPC1MAPTALDH1A1KMT2AMEN1
SCHEMBL6904411 0.72 KDM4E (0.40) MAPTALDH1A1KMT2ARXFP1KDM4E
SCHEMBL29354675 0.70 MAPT (0.43) NPC1MAPTALDH1A1KMT2ARXFP1
SCHEMBL10974102 0.70 NPC1 (0.43) NPC1MAPTALDH1A1KMT2ARXFP1
SCHEMBL5716973 0.70 ALOX5 (0.58) NPC1RXFP1GABRA1GABRB2
SCHEMBL7010787 0.68 ALOX5 (0.56) NPC1MAPTALDH1A1KMT2AMEN1
SCHEMBL6714654 0.68 IDO1 (0.39) ALDH1A1KDM4E
SCHEMBL1420569 0.67 CYP2D6 (0.47) MAPTLMNAPKMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153163-A2 7-Substituted-1-cyclopropyl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids; 7-substituted-1-cyclopropyl-1,4-dihydro-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acids; their derivatives; and a process for preparing the compounds WARNER-LAMBERT COMPANY (US) 1985-08-28 EP disclosed
EP-0106489-A2 Antibacterial agents WARNER-LAMBERT COMPANY (US) 1984-04-25 EP disclosed