SCHEMBL11024944

SCHEMBL11024944

ClCCCN1CCC(c2cccc(Cl)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.52
DRD3 P35462 3/20 0.52
DRD4 P21917 1/20 0.52
GRM2 Q14416 1/20 0.52
HRH3 Q9Y5N1 5/20 0.50
SIGMAR1 Q99720 3/20 0.49
MEN1 O00255 1/20 0.48
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
KMT2A Q03164 1/20 0.48
CCR5 P51681 1/20 0.47
KCNH2 Q12809 1/20 0.47
LMNA P02545 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11027883 0.91 DRD2 (0.54) DRD2DRD3DRD4GRM2SIGMAR1
SCHEMBL2554214 0.83 SIGMAR1 (0.69) DRD2SIGMAR1MEN1TP53CYP1A2
SCHEMBL11023284 0.81 DRD2 (0.71) DRD2DRD3DRD4SIGMAR1MEN1
Hydrochloric Acid SCHEMBL7255548 0.81 SIGMAR1 (0.67) DRD2SIGMAR1MEN1TP53CYP1A2
SCHEMBL7949583 0.79 DRD2 (0.54) DRD2DRD3DRD4KCNH2
SCHEMBL15748120 0.78 DRD2 (0.57) DRD2DRD3DRD4GRM2TSHR
SCHEMBL10078845 0.78 QDPR (0.53) DRD2DRD3DRD4GRM2SLC6A2
SCHEMBL23739762 0.77 HTR1A (0.46) DRD2DRD3DRD4GRM2HRH3
SCHEMBL7963919 0.77 HSD17B10 (0.53) DRD2DRD3DRD4HRH3
SCHEMBL10265025 0.76 DRD2 (0.47) DRD2DRD3DRD4GRM2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0040793-B1 NOVEL QUINAZOLINE-DIONE COMPOUNDS, PROCESS FOR PRODUCTION THEREOF AND PHARMACEUTICAL USE THEREOF Ishikawa, Masayuki (JP) 1985-08-28 EP disclosed
US-4405623-A HYPOTENSIVE AGENTS, VASODILATORS MASAYUKI ISHIKAWA (JP) 1983-09-20 US disclosed
EP-0040793-A1 Novel quinazoline-dione compounds, process for production thereof and pharmaceutical use thereof Ishikawa, Masayuki (JP) 1981-12-02 EP disclosed