SCHEMBL11031350

SCHEMBL11031350

CC(O)(C(=O)N(c1ccc([N+](=O)[O-])c(Cl)c1)N(C(=O)C(C)(O)C(F)(F)F)c1ccc(C#N)c(C#N)c1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.38
NR1H3 Q13133 2/20 0.38
VCAM1 P19320 3/20 0.38
PDK1 Q15118 4/20 0.38
PDK2 Q15119 4/20 0.38
PDK3 Q15120 4/20 0.38
PDK4 Q16654 4/20 0.38
AR P10275 4/20 0.38
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11031351 0.78 ABCC9 (0.53) PDK1PDK2PDK3PDK4AR
SCHEMBL10979529 0.68 MAPT (0.40) NR1H2NR1H3PDK1PDK2PDK3
SCHEMBL10975838 0.66 ABCC9 (0.64) PDK1PDK2PDK3PDK4AR
SCHEMBL11031347 0.65 AR (0.36) VCAM1PDK1PDK2PDK3PDK4
SCHEMBL7526150 0.63 MAPT (0.66) VCAM1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL3725092 0.63 TSHR (0.50) VCAM1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL7642508 0.63 VCAM1 (0.58) VCAM1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL10602642 0.63 MAPT (0.60) VCAM1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL5692532 0.62 PGR (0.43) VCAM1CYP3A4MAPTMAPK1
SCHEMBL7786423 0.62 AR (0.47) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002892-B1 AMIDE DERIVATIVES, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL OR VETERINARY COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-02-06 EP claimed