SCHEMBL11043785

SCHEMBL11043785

CCOC(=O)N1CCC2(CC1)C(=O)NCN2c1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 6/20 0.56
PLD2 O14939 5/20 0.56
OPRK1 P41145 9/20 0.56
HTR2C P28335 4/20 0.54
HTR1A P08908 3/20 0.54
SLC6A3 Q01959 3/20 0.54
ADORA3 P0DMS8 2/20 0.54
OPRM1 P35372 7/20 0.52
AVPR1A P37288 3/20 0.52
HTR7 P34969 3/20 0.52
DRD3 P35462 3/20 0.52
CYP1A2 P05177 2/20 0.52
ADRB1 P08588 2/20 0.52
ADRA2A P08913 2/20 0.52
CYP2D6 P10635 2/20 0.52
DRD2 P14416 2/20 0.52
ADRA2B P18089 2/20 0.52
ADRA2C P18825 2/20 0.52
DRD4 P21917 2/20 0.52
HTR2A P28223 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL318264 0.86 OPRK1 (0.72) PLD1PLD2OPRK1HTR2CHTR1A
SCHEMBL318440 0.85 CCR5 (0.62) PLD1PLD2OPRK1HTR2CHTR1A
SCHEMBL9998386 0.83 OPRM1 (0.60) PLD1PLD2OPRK1HTR2CHTR1A
SCHEMBL3899374 0.81 PLD2 (0.62) PLD1PLD2OPRK1HTR2CHTR1A
SCHEMBL11046747 0.80 DRD2 (0.55) OPRK1OPRM1DRD3DRD2DRD4
SCHEMBL14123322 0.78 BDKRB2 (0.47) OPRK1OPRM1DRD3DRD2DRD4
SCHEMBL318741 0.77 OPRK1 (0.83) OPRK1HTR2CHTR1ASLC6A3ADORA3
SCHEMBL3899569 0.76 OPRM1 (0.57) PLD1PLD2OPRK1HTR2CHTR1A
SCHEMBL15494151 0.76 OPRM1 (0.60) PLD1OPRK1HTR2CHTR1ASLC6A3
SCHEMBL21688364 0.75 OPRM1 (0.56) PLD1PLD2OPRK1HTR2CHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0035902-B1 1-(4-ARYL-CYCLOHEXYL)PIPERIDINE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1984-10-31 EP disclosed
US-4329353-A ANTIEMETIC AND NEUROLEPTIC AGENTS JANSSEN PHARMACEUTICA, N.V. (BE) 1982-05-11 US disclosed
EP-0035902-A1 1-(4-Aryl-cyclohexyl)piperidine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1981-09-16 EP disclosed