SCHEMBL11053236

SCHEMBL11053236

Cc1cccc(Br)c1-n1cnc(N(C)C)nc1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 4/20 0.38
ALDH1A1 P00352 5/20 0.33
CYP1A2 P05177 5/20 0.33
CASP1 P29466 5/20 0.33
CASP7 P55210 5/20 0.33
HSD17B10 Q99714 4/20 0.33
HPGD P15428 3/20 0.33
MAPK1 P28482 2/20 0.33
MEN1 O00255 2/20 0.33
CYP3A4 P08684 2/20 0.33
KMT2A Q03164 2/20 0.33
MAT2A P31153 1/20 0.33
TSHR P16473 1/20 0.33
HIF1A Q16665 2/20 0.32
TP53 P04637 1/20 0.32
GLA P06280 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CYP2D6 P10635 1/20 0.31
DYRK1A Q13627 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056926 0.90 HCAR1 (0.46) HCAR1ALDH1A1CYP1A2CASP1CASP7
Hydrochloric Acid SCHEMBL11056262 0.89 HCAR1 (0.44) HCAR1ALDH1A1CYP1A2CASP1CASP7
SCHEMBL11055971 0.88 HCAR1 (0.36) HCAR1CYP1A2MAT2ACHRNA7
SCHEMBL11059289 0.87 HCAR1 (0.36) HCAR1CHRNA7
SCHEMBL11060207 0.84 HCAR1 (0.38) HCAR1ALDH1A1CYP1A2CASP1CASP7
SCHEMBL11056476 0.81 HCAR1 (0.40) HCAR1ALDH1A1CYP3A4KMT2ACYP2C9
SCHEMBL11057683 0.80 MAPK14 (0.34) HCAR1CYP1A2MAPK1MEN1KMT2A
SCHEMBL10541722 0.79 HCAR1 (0.43) HCAR1ALDH1A1MEN1KMT2ACHRNA7
SCHEMBL11054879 0.78 HCAR1 (0.38) HCAR1CHRNA7PDE7AWEE1
SCHEMBL11052478 0.78 TDP2 (0.33) ALDH1A1CYP1A2CASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed