SCHEMBL11054647

SCHEMBL11054647

CCNc1ncn(-c2c(C)cccc2C)c(=S)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.37
USP2 O75604 7/20 0.35
ALDH1A1 P00352 7/20 0.35
CYP1A2 P05177 7/20 0.35
HSD17B10 Q99714 7/20 0.35
CASP1 P29466 6/20 0.35
CASP7 P55210 6/20 0.35
GLA P06280 5/20 0.35
CYP2D6 P10635 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
TSHR P16473 2/20 0.35
MAPK1 P28482 2/20 0.35
CLK4 Q9HAZ1 2/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CCND2 P30279 1/20 0.35
CCND3 P30281 1/20 0.35
HPGD P15428 3/20 0.34
CYP2C19 P33261 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11053291 0.89 HCAR1 (0.35) HCAR1MEN1KMT2AEGFRFGFR1
SCHEMBL11057004 0.85 LCK (0.43) ALDH1A1CYP1A2HSD17B10CYP2D6TSHR
SCHEMBL11054993 0.84 KCNH2 (0.38) USP2ALDH1A1CYP1A2HSD17B10CASP1
SCHEMBL11050195 0.84 HCAR1 (0.39) HCAR1EGFRFGFR1CHRNA7
SCHEMBL11052901 0.83 HCAR1 (0.43) HCAR1USP2ALDH1A1CYP1A2HSD17B10
Hydrochloric Acid SCHEMBL11343420 0.82 HCAR1 (0.42) HCAR1USP2ALDH1A1CYP1A2HSD17B10
SCHEMBL11058209 0.81 HCAR1 (0.38) HCAR1ALDH1A1KMT2AMAPK1GAA
SCHEMBL11061839 0.80 HCAR1 (0.37) HCAR1CYP1A2KMT2ACDK4CCND1
SCHEMBL11053099 0.80 HCAR1 (0.37) HCAR1ALDH1A1MEN1KMT2ACDK4
SCHEMBL11056523 0.79 MEN1 (0.33) HCAR1CYP1A2CYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed