SCHEMBL11053291

SCHEMBL11053291

CCCNc1ncn(-c2c(C)cccc2C)c(=S)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.35
ELANE P08246 1/20 0.35
SLC2A1 P11166 1/20 0.34
FGFR1 P11362 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
MKNK1 Q9BUB5 3/20 0.32
MKNK2 Q9HBH9 3/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
MERTK Q12866 1/20 0.31
LMNA P02545 2/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
APP P05067 2/20 0.31
BCHE P06276 2/20 0.31
ACHE P22303 2/20 0.31
CHRNA7 P36544 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11054647 0.89 HCAR1 (0.37) HCAR1ELANEFGFR1HTR1AADRA1D
SCHEMBL11059493 0.84 HCAR1 (0.41) HCAR1ELANESLC2A1FGFR1HTR1A
SCHEMBL11057004 0.83 LCK (0.43) ELANELMNAMAPTLCK
SCHEMBL11050195 0.81 HCAR1 (0.39) HCAR1FGFR1CHRNA7EGFR
SCHEMBL11058209 0.79 HCAR1 (0.38) HCAR1LMNAMAPTNPSR1CHRNA7
SCHEMBL11056389 0.78 ELANE (0.38) HCAR1ELANESLC2A1FGFR1LMNA
SCHEMBL11053099 0.78 HCAR1 (0.37) HCAR1ELANEFGFR1CHRNA7MEN1
SCHEMBL11061839 0.78 HCAR1 (0.37) HCAR1CHRNA7KMT2A
SCHEMBL11056591 0.77 KCNH3 (0.39) ELANEFGFR1MAPTNPSR1EGFR
SCHEMBL11057671 0.77 KMT2A (0.42) ELANEFGFR1LMNAMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed