SCHEMBL11058209

SCHEMBL11058209

Cc1cccc(C)c1Nc1ncn(-c2c(C)cccc2C)c(=S)n1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.38
SRC P12931 3/20 0.35
GAA P10253 2/20 0.34
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CHRNA7 P36544 7/20 0.34
LCK P06239 2/20 0.34
LMNA P02545 1/20 0.33
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32
CRHR1 P34998 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11061669 0.86 WEE1 (0.44) SRCMAPTMAPK1KMT2ACHRNA7
SCHEMBL11050195 0.85 HCAR1 (0.39) HCAR1SRCCHRNA7
SCHEMBL11053933 0.82 HCAR1 (0.43) HCAR1SRCGAAMAPTMAPK1
SCHEMBL11053099 0.81 HCAR1 (0.37) HCAR1GAAKMT2ACHRNA7LCK
SCHEMBL11061839 0.81 HCAR1 (0.37) HCAR1KMT2ASMN1; SMN2CHRNA7
SCHEMBL11054647 0.81 HCAR1 (0.37) HCAR1GAAMAPK1KMT2ASMN1; SMN2
SCHEMBL11053291 0.79 HCAR1 (0.35) HCAR1MAPTKMT2ANPSR1CHRNA7
SCHEMBL11057546 0.79 KDM4E (0.41) GAASMN1; SMN2LMNA
SCHEMBL11057004 0.78 LCK (0.43) GAAMAPTMAPK1SMN1; SMN2L3MBTL1
SCHEMBL11057092 0.76 CHRNA7 (0.44) HCAR1SRCCHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed