SCHEMBL11065008

SCHEMBL11065008

Brc1nc(Cc2ccccc2)cs1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.44
HDAC1 Q13547 5/20 0.44
HDAC6 Q9UBN7 5/20 0.44
CALM1 P0DP23 1/20 0.42
LTA4H P09960 1/20 0.42
HDAC8 Q9BY41 1/20 0.41
C1S P09871 1/20 0.41
ALDH1A1 P00352 2/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
AOC3 Q16853 1/20 0.38
BRD4 O60885 1/20 0.37
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11260478 0.86 SLC6A4 (0.42) NOS1HDAC1HDAC6LTA4HHDAC8
SCHEMBL11261522 0.82 HTR6 (0.44) HDAC1HDAC6ALDH1A1SMN1; SMN2TDP1
SCHEMBL11259748 0.82 HDAC1 (0.34) NOS1HDAC1HDAC6LTA4HHDAC8
SCHEMBL28759152 0.80 HDAC1 (0.59) NOS1HDAC1HDAC6CALM1LTA4H
SCHEMBL2705651 0.79 HDAC1 (0.48) NOS1HDAC1HDAC6CALM1LTA4H
SCHEMBL25427585 0.78 SLC6A3 (0.50) NOS1HDAC1HDAC6CALM1LTA4H
SCHEMBL2263697 0.78 SLC6A3 (0.53) NOS1C1SALDH1A1SMN1; SMN2
SCHEMBL1915556 0.78 NOS1 (0.71) NOS1LTA4HALDH1A1RAB9ASMN1; SMN2
SCHEMBL6377492 0.78 NOS1 (0.43) NOS1HDAC1HDAC6CALM1LTA4H
SCHEMBL28177852 0.78 DRD2 (0.61) C1SALDH1A1RAB9ASMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4479952-A 1-(4-benzyl-2-thiazolyl) piperazine; antiinflammatory; immunomodulator SCIENCE UNION ET CIE (FR) 1984-10-30 US disclosed