SCHEMBL11065024

SCHEMBL11065024

COc1nc(C)nc(Cl)c1NC(N)=S

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
HTR1A P08908 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
HRH2 P25021 1/20 0.46
CYP2C19 P33261 1/20 0.46
ADRA1A P35348 1/20 0.46
NISCH Q9Y2I1 1/20 0.46
TDP1 Q9NUW8 2/20 0.45
ALOX15 P16050 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
HTT P42858 2/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10957823 0.88 ALDH1A1 (0.37) LMNAHTR1AADRA2AADRA2BADRA2C
SCHEMBL11058765 0.78 ADORA3 (0.34) LMNAHTR1AADRA2AADRA2BADRA2C
SCHEMBL11061561 0.77 HTT (0.33) TDP1HTTALDH1A1KMT2A
SCHEMBL11062612 0.74 HTT (0.35) CYP2C19TDP1HTTALDH1A1KMT2A
SCHEMBL11059523 0.72 ALDH1A1 (0.34) TDP1HTTALDH1A1KMT2A
SCHEMBL11069778 0.71 ALDH1A1 (0.36) TDP1HTTALDH1A1KMT2A
SCHEMBL29261699 0.71 CCR4 (0.33) LMNACYP2C19HTTALDH1A1KMT2A
SCHEMBL11055958 0.70 HTT (0.40) CYP2C19TDP1HTTALDH1A1KMT2A
SCHEMBL11058164 0.69 ALDH1A1 (0.41) LMNATDP1HTTALDH1A1KMT2A
SCHEMBL11058685 0.68 L3MBTL1 (0.40) LMNACYP2C19HTTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4434167-A Pyrimidyl thioureas useful for the treatment of hypertension and hyperlipidemia BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-02-28 US disclosed