SCHEMBL11069100

SCHEMBL11069100

CC(C)N1CC(COc2cccc3c(=O)n(CC4CN(C(C)C)C(=O)O4)ccc23)OC1=O

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 1/20 0.42
GRM2 Q14416 4/20 0.38
KDM4E B2RXH2 11/20 0.37
RXFP1 Q9HBX9 1/20 0.36
ALDH1A1 P00352 4/20 0.36
TSHR P16473 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTT P42858 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9225959 0.82 PDK1 (0.46) HTR2BGRM2KDM4EALDH1A1TSHR
SCHEMBL9225971 0.82 PDK1 (0.46) HTR2BGRM2KDM4EALDH1A1TSHR
SCHEMBL11071694 0.81 PARP1 (0.44) HTR2BGRM2KDM4EALDH1A1HSD17B10
SCHEMBL11067676 0.78 GRM2 (0.39) HTR2BGRM2
SCHEMBL11060976 0.78 GRM2 (0.43) HTR2BGRM2
SCHEMBL11067481 0.77 GRM2 (0.38) HTR2BGRM2
SCHEMBL11220571 0.76 HTR1A (0.45) KDM4EALDH1A1TSHR
SCHEMBL11875374 0.76 HTR2B (0.47) HTR2BGRM2
SCHEMBL11068306 0.74 ADRB2 (0.44) HTR2BGRM2NPC1
SCHEMBL11071828 0.73 HTR2B (0.37) HTR2BGRM2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4473501-A HYPOTENSIVES G. D. SEARLE & CO. (US) 1984-09-25 US disclosed
EP-0064294-A1 1,5-Substituted isoquinoline derivatives G.D. Searle & Co. (US) 1982-11-10 EP disclosed