SCHEMBL9225971

SCHEMBL9225971

CC(C)N1CC(COc2cccc3ccccc23)OC1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.46
HTR2B P41595 4/20 0.45
GRM2 Q14416 8/20 0.45
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HTR1B P28222 2/20 0.40
TSHR P16473 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP1A2 P05177 3/20 0.40
ADRB2 P07550 3/20 0.40
ADRB1 P08588 3/20 0.40
CYP2D6 P10635 3/20 0.40
SLC6A4 P31645 3/20 0.40
SIGMAR1 Q99720 3/20 0.40
NR2E1 Q9Y466 3/20 0.40
ADRB3 P13945 2/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9225959 1.00 PDK1 (0.46) PDK1HTR2BGRM2ALDH1A1KDM4E
SCHEMBL11068306 0.87 ADRB2 (0.44) HTR2BGRM2ADRB2ADRB1ADRB3
SCHEMBL11071694 0.85 PARP1 (0.44) HTR2BGRM2ALDH1A1KDM4EKMT2A
SCHEMBL11071828 0.85 HTR2B (0.37) PDK1HTR2BGRM2ALDH1A1KDM4E
SCHEMBL11875374 0.84 HTR2B (0.47) HTR2BGRM2L3MBTL1ADRA2CMAPK1
SCHEMBL11067676 0.82 GRM2 (0.39) HTR2BGRM2L3MBTL1MAPK1
SCHEMBL11060976 0.82 GRM2 (0.43) HTR2BGRM2L3MBTL1MAPK1
SCHEMBL11220571 0.82 HTR1A (0.45) ALDH1A1KDM4EMEN1KMT2AHTR1B
SCHEMBL11069100 0.82 HTR2B (0.42) HTR2BGRM2ALDH1A1KDM4ETSHR
SCHEMBL14168333 0.81 HTR2B (0.43) HTR2BGRM2ALDH1A1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647634-A1 Method of preparing a heterocyclic intermediate for the production of optically active aryloxy-substituted vicinal aminoalcohols DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1995-04-12 EP disclosed
EP-0647633-A1 Method of preparing a heterocyclic intermediate for the production of optically active aryloxysubstituted vicinal aminoalcohols DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1995-04-12 EP disclosed
EP-0008711-B1 A METHOD OF PREPARING A 2-HYDROXY-3-ISOPROPYL OR A 2-HYDROXY-3-TERT-BUTYLAMINOPROPYL AROMATIC ETHER SMITHKLINE BECKMAN CORPORATION (US) 1981-11-04 EP disclosed
EP-0008711-A1 A method of preparing a 2-hydroxy-3-isopropyl or a 2-hydroxy-3-tert-butylaminopropyl aromatic ether SMITHKLINE BECKMAN CORPORATION (US) 1980-03-19 EP disclosed