SCHEMBL11076008

SCHEMBL11076008

CN(C)Cc1ccc(CC(C=O)C(=O)O)cn1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 9/20 0.36
CPA1 P15085 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
MCHR1 Q99705 4/20 0.32
S1PR2 O95136 1/20 0.32
S1PR3 Q99500 1/20 0.32
CPB1 P15086 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080782 0.85 CPB2 (0.38) CPB2HDAC3HDAC6MEN1KMT2A
SCHEMBL11022295 0.79 TSHR (0.46) CPB2CPA1HDAC6MEN1KMT2A
SCHEMBL11078876 0.73 ALDH1A1 (0.42) MEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL11076247 0.71 P4HTM (0.54) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL7005064 0.70 GRN (0.39) MEN1KMT2AALDH1A1MAPTMAPK1
SCHEMBL9900895 0.70 LDHA (0.36) CPB2CPA1
SCHEMBL11955565 0.69 HRH3 (0.47) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL10740513 0.69 CPB2 (0.40) CPB2CPB1
SCHEMBL1713633 0.68 HCAR3 (0.55) KDM4EALDH1A1MAPTCYP2C19
SCHEMBL7395620 0.68 P4HTM (0.57) HDAC3HDAC6MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0039989-B1 PYRIMIDONE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-08-29 EP disclosed
US-4388317-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-06-14 US disclosed
EP-0039989-A1 Pyrimidone derivatives, processes for their preparation and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-11-18 EP disclosed