SCHEMBL11078097

SCHEMBL11078097

NC(=O)CC(CC(N)=O)c1cc(Br)cc(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
EPHX1 P07099 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP2C19 P33261 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
PKM P14618 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PARP1 P09874 1/20 0.31
IKBKB O14920 1/20 0.31
USP2 O75604 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31
MAPK10 P53779 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11079107 0.81 PARP1 (0.47) ALDH1A1SMN1; SMN2L3MBTL1CYP1A2CYP2D6
SCHEMBL7417348 0.80 EPHX1 (0.33) EPHX1SMN1; SMN2L3MBTL1CYP2C19MEN1
SCHEMBL11084494 0.79 ALOX5 (0.46) ALDH1A1EPHX1SMN1; SMN2MEN1KMT2A
SCHEMBL11084618 0.75 ITGB3 (0.40) ALDH1A1CYP2C19MEN1KMT2ACYP1A2
SCHEMBL11079409 0.75 CES2 (0.42) ALDH1A1EPHX1L3MBTL1
SCHEMBL11083231 0.70 HTR2A (0.37)
SCHEMBL9105247 0.70 ALDH1A1 (0.63) ALDH1A1EPHX1SMN1; SMN2L3MBTL1CYP2C19
SCHEMBL11077388 0.69 KMT2A (0.34) EPHX1SMN1; SMN2MEN1KMT2AALOX15
SCHEMBL11079401 0.69 SMN1; SMN2 (0.37) SMN1; SMN2MEN1KMT2APARP1ALOX15
SCHEMBL19067137 0.69 KMT2A (0.42) EPHX1SMN1; SMN2CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed