SCHEMBL11079956

SCHEMBL11079956

CNc1nc(Nc2ccc(Cl)cc2)no1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.43
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
GAA P10253 2/20 0.41
ADORA3 P0DMS8 1/20 0.41
SLC6A2 P23975 1/20 0.41
PDE4A P27815 1/20 0.41
KDR P35968 1/20 0.41
GFER P55789 1/20 0.41
KCNH3 Q9ULD8 1/20 0.41
NR1I2 O75469 1/20 0.41
AHR P35869 1/20 0.41
SCN9A Q15858 2/20 0.41
TNNI3K Q59H18 1/20 0.39
LMNA P02545 1/20 0.39
JAK2 O60674 1/20 0.39
LRRK2 Q5S007 1/20 0.39
ALDH1A1 P00352 3/20 0.38
NPC1 O15118 2/20 0.38
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11089831 0.83 NPY5R (0.41) GAAKDRJAK2LRRK2NPC1
SCHEMBL11080475 0.77 MEN1 (0.53) POLBMEN1KMT2AGAAADORA3
SCHEMBL11080739 0.75 C1R (0.38) MEN1KMT2AGAALMNAJAK2
SCHEMBL11256388 0.75 NPY5R (0.38) POLBMEN1KMT2AJAK2LRRK2
SCHEMBL14869704 0.74 LMNA (0.65) POLBMEN1KMT2AGAAADORA3
SCHEMBL11082598 0.74 TSHR (0.51) KMT2ALRRK2ALDH1A1NPC1MAPT
SCHEMBL11630110 0.71 KCNH3 (0.59) POLBMEN1KMT2AGAAADORA3
SCHEMBL11788144 0.70 LMNA (0.74) POLBMEN1KMT2AGAAKCNH3
SCHEMBL4416547 0.70 CASP3 (0.62) MEN1KMT2AGAAADORA3SLC6A2
SCHEMBL17377367 0.69 MAPT (0.48) POLBMEN1KMT2AGAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US claimed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP claimed
US-4446142-A HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-05-01 US disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed
EP-0044266-A2 Substituted 3,5-diamino-1,2,4-oxadiazoles and 3,5-diamino-1,2,4-thiadiazoles, their preparation and pharmaceutical compositions containing them Beiersdorf Aktiengesellschaft (DE) 1982-01-20 EP disclosed