SCHEMBL11087355

SCHEMBL11087355

CC1CCc2ncc(-c3ccccc3)c(=O)n21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
CYP1A2 P05177 5/20 0.37
TSHR P16473 5/20 0.37
CYP2C9 P11712 4/20 0.37
CYP2C19 P33261 4/20 0.37
MAPK1 P28482 3/20 0.37
HPGD P15428 3/20 0.37
HSD17B10 Q99714 3/20 0.37
ALOX15 P16050 2/20 0.37
CASP1 P29466 2/20 0.37
CASP7 P55210 2/20 0.37
GLA P06280 1/20 0.37
HIF1A Q16665 1/20 0.37
USP30 Q70CQ3 1/20 0.37
MAP3K5 Q99683 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
RAB9A P51151 2/20 0.35
CYP3A4 P08684 3/20 0.34
USP2 O75604 2/20 0.34
PTGS2 P35354 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11090649 0.75 MAP3K5 (0.33) ALDH1A1CYP1A2CYP2C9CYP2C19MAPK1
SCHEMBL11084126 0.75 CYP1A2 (0.34) ALDH1A1CYP1A2TSHRCYP2C9CYP2C19
SCHEMBL11084986 0.75 ALDH1A1 (0.46) ALDH1A1CYP1A2TSHRCYP2C9CYP2C19
SCHEMBL11084988 0.75 ALDH1A1 (0.46) ALDH1A1CYP1A2TSHRCYP2C9CYP2C19
SCHEMBL11086999 0.74 CHEK1 (0.38) ALDH1A1CYP1A2HPGDHIF1ASMN1; SMN2
SCHEMBL12946456 0.73 RAB9A (0.44) ALDH1A1CYP1A2CYP2C19HPGDSMN1; SMN2
SCHEMBL12747498 0.72 KAT2B (0.35) CYP1A2CYP2C9SMN1; SMN2RAB9ANPC1
SCHEMBL15160572 0.71 ALOX15 (0.52) ALDH1A1CYP1A2TSHRHSD17B10ALOX15
SCHEMBL11088686 0.70 ADORA2A (0.38) ALDH1A1MAPK1HPGDHSD17B10CASP1
SCHEMBL11088861 0.70 NNMT (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4482557-A 3-Substituted-2-oxo-tetrahydro-pyrrol[1,2-a]pyrimidines having digitalis-like activity CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1984-11-13 US disclosed
US-4367229-A 3-Substituted-tetrahydro-pyrrolo[1,2-a]pyrimidines and pharmaceutical compositions CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1983-01-04 US disclosed