SCHEMBL11088686

SCHEMBL11088686

CC1CCc2nc(=O)c(-c3ccccc3)cn21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.38
P2RX7 Q99572 1/20 0.36
ALDH1A1 P00352 4/20 0.35
WDR5 P61964 2/20 0.35
SRC P12931 3/20 0.35
MAP3K5 Q99683 1/20 0.34
BRD4 O60885 1/20 0.34
ABL1 P00519 2/20 0.33
EGFR P00533 2/20 0.33
ABL2 P42684 2/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
LMNA P02545 2/20 0.33
RAB9A P51151 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11087486 0.71 WDR5 (0.64) ALDH1A1WDR5KDM4ENPC1LMNA
SCHEMBL11087355 0.70 ALDH1A1 (0.37) ALDH1A1SRCMAP3K5BRD4NPC1
SCHEMBL11192535 0.69 WDR5 (0.56) ALDH1A1WDR5KDM4ENPC1LMNA
SCHEMBL11093001 0.69 KDM4E (0.37) P2RX7KDM4ELMNASMN1; SMN2
SCHEMBL22854685 0.69
SCHEMBL24880388 0.67 HTR2A (0.30)
SCHEMBL22833685 0.67
SCHEMBL16772981 0.67 SMN1; SMN2 (0.42) ALDH1A1WDR5MAP3K5KDM4ENPC1
SCHEMBL15160572 0.63 ALOX15 (0.52) ALDH1A1KDM4ELMNAHSD17B10MAPT
SCHEMBL11748346 0.59 CYP2E1 (0.45) ALDH1A1SRCBRD4KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4482557-A 3-Substituted-2-oxo-tetrahydro-pyrrol[1,2-a]pyrimidines having digitalis-like activity CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1984-11-13 US disclosed
US-4367229-A 3-Substituted-tetrahydro-pyrrolo[1,2-a]pyrimidines and pharmaceutical compositions CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1983-01-04 US disclosed