SCHEMBL11084126

SCHEMBL11084126

CC1CCC(Br)(Br)c2ncc(-c3ccccc3)c(=O)n21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.34
ALDH1A1 P00352 5/20 0.34
CYP2C9 P11712 4/20 0.34
TSHR P16473 4/20 0.34
CYP2C19 P33261 4/20 0.34
HPGD P15428 4/20 0.34
HSD17B10 Q99714 4/20 0.34
MAPK1 P28482 3/20 0.34
CASP1 P29466 3/20 0.34
CASP7 P55210 3/20 0.34
ALOX15 P16050 2/20 0.34
HIF1A Q16665 2/20 0.34
GLA P06280 1/20 0.34
LYN P07948 6/20 0.33
SRC P12931 4/20 0.33
HRH3 Q9Y5N1 1/20 0.32
CYP3A4 P08684 3/20 0.32
USP30 Q70CQ3 1/20 0.32
BRD4 O60885 1/20 0.31
ATAD2 Q6PL18 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11087355 0.75 ALDH1A1 (0.37) CYP1A2ALDH1A1CYP2C9TSHRCYP2C19
SCHEMBL11084988 0.65 ALDH1A1 (0.46) CYP1A2ALDH1A1CYP2C9TSHRCYP2C19
SCHEMBL11084986 0.65 ALDH1A1 (0.46) CYP1A2ALDH1A1CYP2C9TSHRCYP2C19
SCHEMBL11270993 0.59 KDM4E (0.47) ALDH1A1HSD17B10MAPK1ALOX15BRD4
SCHEMBL11096181 0.56 ALDH1A1 (0.54) CYP1A2ALDH1A1CYP2C9CYP2C19HPGD
SCHEMBL29126016 0.56 BRD9 (0.51) CYP1A2ALDH1A1TSHRCYP3A4BRD4
SCHEMBL2834048 0.55 GABRA1 (0.44) CYP1A2ALDH1A1CYP2C19HPGDHSD17B10
SCHEMBL11088686 0.54 ADORA2A (0.38) ALDH1A1HPGDHSD17B10MAPK1CASP1
SCHEMBL11177118 0.54 ALDH1A1 (0.61) CYP1A2ALDH1A1HPGDHSD17B10MAPK1
SCHEMBL11575773 0.52 KDM4E (0.54) ALDH1A1HSD17B10MAPK1GLAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4456752-A REACTING A HYDRAZINE WITH DIHALOGEN SUBSTITUTED PYRIDO(1,2-A)PYRIMIDINE CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA R.T. (HU) 1984-06-26 US disclosed