SCHEMBL11087486

SCHEMBL11087486

O=c1nc2n(cc1-c1ccccc1)CCC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 9/20 0.64
ALDH1A1 P00352 4/20 0.64
NPC1 O15118 5/20 0.59
RAB9A P51151 5/20 0.59
LMNA P02545 3/20 0.59
HTT P42858 2/20 0.59
KDM4E B2RXH2 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.48
TP53 P04637 1/20 0.48
HSD17B10 Q99714 2/20 0.46
PTGS2 P35354 3/20 0.44
ALOX5 P09917 2/20 0.44
KMT2A Q03164 2/20 0.43
MAPT P10636 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
PTGS1 P23219 1/20 0.43
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42
BCHE P06276 1/20 0.42
CFTR P13569 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11192535 0.94 WDR5 (0.56) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL989261 0.78 WDR5 (1.00) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL4839937 0.73 WDR5 (0.90) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL11087009 0.72 WDR5 (0.47) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL17767605 0.70 WDR5 (0.56) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL11097275 0.70 WDR5 (0.46) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL7380842 0.70 WDR5 (0.65) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL9532243 0.69 PTGS2 (0.75) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL18007543 0.69
SCHEMBL11096181 0.67 ALDH1A1 (0.54) WDR5ALDH1A1NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4482557-A 3-Substituted-2-oxo-tetrahydro-pyrrol[1,2-a]pyrimidines having digitalis-like activity CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1984-11-13 US disclosed
US-4367229-A 3-Substituted-tetrahydro-pyrrolo[1,2-a]pyrimidines and pharmaceutical compositions CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1983-01-04 US disclosed