SCHEMBL11096161

SCHEMBL11096161

COc1cc(NC=O)c(Cl)cc1NC(=O)C1CC2CCC(C1)N2CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 9/20 0.51
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
DRD3 P35462 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
OPRK1 P41145 1/20 0.43
KCNH2 Q12809 1/20 0.43
MAPK1 P28482 1/20 0.42
TSHR P16473 1/20 0.42
CHRNA7 P36544 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11097324 0.92 DRD4 (0.48) DRD4HPGDDRD3OPRM1OPRK1
SCHEMBL11096503 0.86 DRD2 (0.52) DRD4HPGDSMN1; SMN2DRD3OPRK1
SCHEMBL11093528 0.85 CXCR6 (0.47) DRD4DRD3TSHR
SCHEMBL11099467 0.85 TSHR (0.44) DRD4DRD3TSHR
SCHEMBL11346054 0.84 MAPK1 (0.60) DRD4SMN1; SMN2MAPK1
SCHEMBL11094396 0.84 SIGMAR1 (0.46) DRD4DRD3OPRM1OPRD1OPRK1
SCHEMBL11100788 0.84 TSHR (0.43) DRD4SMN1; SMN2OPRM1OPRD1TSHR
SCHEMBL11270864 0.84 CXCR4 (0.46) DRD4DRD3TSHR
SCHEMBL11097362 0.83 TSHR (0.43) DRD4DRD3TSHR
SCHEMBL11095214 0.82 UBE2M (0.44) DRD4HPGDSMN1; SMN2DRD3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-B1 ANILINE DERIVATIVES BEECHAM GROUP PLC (GB) 1984-03-07 EP disclosed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed